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METHOD OF SYNTHESIS OF NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS

机译:含氮杂环化合物或其药学上可接受的盐的合成方法

摘要

FIELD: organic chemistry. SUBSTANCE: method involves the synthesis of new heterocyclic nitrogen-containing compounds of the formula (I) where radicals R1-R4 have different meanings; X - CH2 , or their pharmaceutically acceptable salts. Reagent 1: compound of the formula (II) where R - H. Reagent 2: R2-Y. Synthesized compounds are used in medicine. EFFECT: improved method of synthesis of compounds indicated above. 1 tbl
机译:领域:有机化学。物质:该方法涉及合成新的式(I)的杂环含氮化合物,其中基团R 1 -R 4 具有不同的含义; X-CH 2 或其可药用盐。试剂1:式(II)的化合物,其中R-H。试剂2:R 2 -Y。合成的化合物用于医学。效果:改进了上述化合物的合成方法。 1汤匙

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