首页> 外国专利> 5 - PHENYL - PYRAZOLO 1,5-a PYRIMIDINE - 3 - CARBOXYLIC ACID (3 - SULFONYL - PHENYL) - AMIDE DERIVATIVES, THEIR MANUFACTURE AND USE THEREOF IN THE PREPARATION OF MEDICAMENTS FOR THE TREATMENT OR PREVENTION OF ACUTE OR CHRONIC NEUROLOGICAL DISORDERS

5 - PHENYL - PYRAZOLO 1,5-a PYRIMIDINE - 3 - CARBOXYLIC ACID (3 - SULFONYL - PHENYL) - AMIDE DERIVATIVES, THEIR MANUFACTURE AND USE THEREOF IN THE PREPARATION OF MEDICAMENTS FOR THE TREATMENT OR PREVENTION OF ACUTE OR CHRONIC NEUROLOGICAL DISORDERS

机译:5-苯基-吡唑并[1,5-a]嘧啶-3-羧酸(3-磺酰基-苯基)-酰胺衍生物,其制备及在制备用于治疗或预防急性或慢性神经疾病的药物中

摘要

The invention relates to compounds of formula (I) wherein RSUP1/SUP, RSUP2/SUP, RSUP3/SUP, RSUP4/SUP, RSUP5 /SUPand p are as defined in the description and to pharmaceutically acceptable salts thereof, to pharmaceutical compositions containing such compounds, to the manufacture of such compounds and compositions, and to methods of treating or preventing acute and/or chronic central nervous system disorders by administering such compounds.
机译:本发明涉及式(I)的化合物,其中R 1 ,R 2 ,R 3 ,R 4 ,R 5 和p如说明书中所定义,及其药学上可接受的盐,含有此类化合物的药物组合物,此类化合物和组合物的制备以及治疗或预防急性和慢性精神病的方法/或通过施用此类化合物来治疗慢性中枢神经系统疾病。

著录项

  • 公开/公告号IL179736A

    专利类型

  • 公开/公告日2010-12-30

    原文格式PDF

  • 申请/专利权人 F. HOFFMANN-LA ROCHE AG;

    申请/专利号IL20060179736

  • 发明设计人

    申请日2006-11-30

  • 分类号C07D487/04;

  • 国家 IL

  • 入库时间 2022-08-21 18:06:25

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