首页> 外国专利> CRYSTALLINE FORM OF (S)-2-(8-((5-CHLOROPYRIMIDIN-2-YL)(METHYL)AMINO)-2-FLUORO-6,7,8,9-TETRAHYDRO-5H-PYRIDO3,2-bINDOL-5-YL)ACETIC ACID AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME

CRYSTALLINE FORM OF (S)-2-(8-((5-CHLOROPYRIMIDIN-2-YL)(METHYL)AMINO)-2-FLUORO-6,7,8,9-TETRAHYDRO-5H-PYRIDO3,2-bINDOL-5-YL)ACETIC ACID AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME

机译:(S)-2-(8-((5-氯代嘧啶-2-基)(甲基)亚氨基)-2-氟-6,7,8,9-四氢-5H-吡咯并[3,2- b]吲哚-5-基)乙酸和组成相同的药物

摘要

The invention relates to a new crystalline form of (S)-2-(8-((5-chloropyrimidin-2-yl)(methyl)amino)-2-fluoro-6,7,8,9-tetrahydro-5H-pyrido[3,2-b]indol-5-yl)acetic acid, pharmaceutical compositions comprising such crystalline form, and the use of this crystalline form as medicaments, especially as CRTH2 (chemoattractant receptor-homologous molecule expressed on Th2 cells) receptor modulators.
机译:本发明涉及(S)-2-(8-((5-氯嘧啶-2-基)(甲基)氨基)-2-氟-6,7,8,9-四氢-5H-的新晶型吡啶并[3,2-b]吲哚-5-基)乙酸,包含这种晶型的药物组合物,以及该晶型作为药物的用途,尤其是作为CRTH2(在Th2细胞上表达的化学吸引剂受体-同源分子)受体调节剂。

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