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机译:通过高通量筛选,晶体学和基于细胞的测定来发现新型BRD4抑制剂
Nanchang Univ Sch Pharm 461 Bayi Rd Nanchang 330006 Jiangxi Peoples R China;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
ShanghaiTech Univ Sch Life Sci &
Technol 100 Haike Rd Shanghai 201210 Peoples R China;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
Nanchang Univ Sch Pharm 461 Bayi Rd Nanchang 330006 Jiangxi Peoples R China;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
Chinese Acad Sci Shanghai Inst Mat Med Drug Discovery &
Design Ctr State Key Lab Drug Res 555;
BRD4 inhibitor; High-throughput screening; Crystallography;
机译:通过高通量筛选,晶体学和基于细胞的测定来发现新型BRD4抑制剂
机译:发现新型三甲氧基环BRD4溴染色蛋白抑制剂:α谱系测定,晶体学和基于细胞的测定
机译:高通量基于细胞的筛选,使用闪烁接近分析法测定肌醇磷酸酶抑制剂
机译:高通量药物发现:由人肾上腺素合成酶PNMT的X射线晶体学基于碎片的筛选
机译:基于细胞的足细胞高通量筛选检测方法的开发。
机译:发现新型三甲氧基环BRD4溴结构域抑制剂:AlphaScreen测定,晶体学和基于细胞的测定
机译:基于高通量的细胞基筛选用于发现肌醇磷酸酶抑制剂的闪烁近距离测定