Synthesis of 3-aryl-2-tert.butylimino-6-p-tolylimino-4-(5-tetra-O-benzoyl-D-glucopyranosyl)-2,3-dihydro-1,3,5-thiadiazine hydrochlorides and their antibacterial and antifungal studies

摘要

Some 3-aryl-2-tert.butylimino-6-p-tolylimino-4-S-tctra-O-bcnzoyl-D-glucopyranosyl-2,3-dihydro-1,3,5-thiadiazines (hydrochlorides) have been prepared by the interaction of 2-(S-tetra-O-benzoyl-D-glucopyranosyl)-l-aryl-5-p-tolyl-2,4-isodithiobiurets and tert.butyl isocyanodichluridc.These compounds show good to moderate antibacterial and antifungal activities.All products are optically active.