首页> 外国专利> NEW SPARTEINE DERIVATIVE,PROCESS FOR THEIR PRODUCTION,PHARMACEUTICAL PRODUCTS CONTAINING THE DERIVATIVE AND PROCESS FOR PRODUCING THE PHARMACEUTICAL PRODUCTS.

NEW SPARTEINE DERIVATIVE,PROCESS FOR THEIR PRODUCTION,PHARMACEUTICAL PRODUCTS CONTAINING THE DERIVATIVE AND PROCESS FOR PRODUCING THE PHARMACEUTICAL PRODUCTS.

机译:新的斯帕汀衍生物,其生产过程,包含该衍生物的药物和生产该药物的过程。

摘要

Disclosed are a novel dimeric sparteine derivative, the 17S,17'S-bissparteine, and its physiologically compatible acid addition salts. Said compounds are produced by dimerization of 17-hydroxy sparteine or 17-dehydrosparteine salts by means of activated magnesium or an alkali metal. Pharmaceutical compositions containing said novel dimeric sparteine derivatives and their preparation are also described.
机译:公开了一种新型的二聚体天冬氨酸衍生物,17S,17′S-双天冬氨酸及其生理相容的酸加成盐。所述化合物通过借助于活化镁或碱金属使17-羟基天冬氨酸或17-脱氢天冬氨酸盐二聚而产生。还描述了包含所述新颖的二聚体天冬氨酸衍生物的药物组合物及其制备。

著录项

  • 公开/公告号JPS57501582A

    专利类型

  • 公开/公告日1982-09-02

    原文格式PDF

  • 申请/专利权人

    申请/专利号JP19810502804

  • 发明设计人

    申请日1981-08-18

  • 分类号A61K31/435;A61P9/06;C07D471/00;C07D471/22;C07D519/00;

  • 国家 JP

  • 入库时间 2022-08-22 14:01:28

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