首页> 外国专利> NOVEL QUINAZOLINE DERIVATIVES, A PHARMACEUTICAL COMPOSITION CONTAINING SUCH DERIVATIVES AS ACTIVE INGREDIENT AND A PROCESS FOR PRODUCING THE QUINAZOLINE DERIVATIVES

NOVEL QUINAZOLINE DERIVATIVES, A PHARMACEUTICAL COMPOSITION CONTAINING SUCH DERIVATIVES AS ACTIVE INGREDIENT AND A PROCESS FOR PRODUCING THE QUINAZOLINE DERIVATIVES

机译:新型喹唑啉衍生物,一种包含这类衍生物作为活性成分的药物组合物,以及制备喹唑啉衍生物的方法

摘要

There are presented novel quinazoline derivatives, namely 2-(4-substituted-carbamoyl-piperazin-1-yl)quinazoline derivatives, 2-(4-substituted-carbamoyl-homopiperazin-1-yl)quinazoline derivatives, 2-(4-substituted-thiocarbamoyl-piperazin-1-yl)quinazoline derivatives and 2-(4-substituted-thiocarbamoyl-piperazin-1-yl)quinazoline derivatives, having excellent antihypertensive activities.
机译:提出了新颖的喹唑啉衍生物,即2-(4-取代的氨基甲酰基-哌嗪-1-基)喹唑啉衍生物,2-(4-取代的氨基甲酰基-高哌嗪-1-基)喹唑啉衍生物,2-(4-取代的) -硫代氨基甲酰基-哌嗪-1-基)喹唑啉衍生物和2-(4-取代-硫代氨基甲酰基-哌嗪-1-基)喹唑啉衍生物,具有优异的降压活性。

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