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Novel quinazoline derivatives, a pharmaceutical composition containing such derivatives as active ingredient and a process for producing the quinazoline derivatives

机译:新型喹唑啉衍生物,含有此类衍生物作为活性成分的药物组合物和制备喹唑啉衍生物的方法

摘要

There are presented novel quinazoline derivatives, namely 2-(4-substituted-carbamoyl-piperazin-1-yl)quinazoline derivatives, 2-(4-substituted-carbamoyl-homopiperazin-1--yl)quinazoline derivatives, 2-(4-substituted-thiocarbamoyl--piperazin-a-yl)quinazoline derivatives and 2-(4-substituted--thiocarbamoyl-piperazin-1-yl)quinazoline derivatives and a process for producing same. In form of pharmaceutical preparation said derivatives exhibit excellent antihypertensive activities.
机译:提出了新颖的喹唑啉衍生物,即2-(4-取代的氨基甲酰基-哌嗪-1-基)喹唑啉衍生物,2-(4-取代的氨基甲酰基-高哌嗪-1-基)喹唑啉衍生物,2-(4-取代的硫代氨基甲酰基-哌嗪-a-基)喹唑啉衍生物和2-(4-取代的硫代氨基甲酰基-哌嗪-1-基)喹唑啉衍生物及其制备方法。在药物制剂的形式中,所述衍生物表现出优异的抗高血压活性。

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