首页> 外国专利> A process for the production of a derivative of Diami-N-acylamino das

A process for the production of a derivative of Diami-N-acylamino das

机译:制备二氨基-N-酰氨基达斯衍生物的方法

摘要

This invention relates to a novel N-acyl acidic amino acid diamide derivative represented by the general formula or a salt thereof: IMAGE wherein each of R1, R2, R3 and R4, which may be the same or different, represents a hydrogen atom or a substituted or unsubstituted alkyl, cycloalkyl, alkenyl or aralkyl group, or R1 and R2 and/or R3 and R4, when taken together with the respective adjacent nitrogen atoms, form a substituted or unsubstituted heterocyclic group; R5 represents a substituted or unsubstituted cycloalkyl, acyl or heterocyclic group; A represents a bond or a substituted or unsubstituted alkylene, alkenylene or alkadienylene group; and n is 1, 2 or 3. Said compound has an anti-ulcer activity which is effective to human beings and animals. This disclosure relates to such a compound, to a process for the production thereof and to an anti-ulcer agent containing the same.
机译:本发明涉及由通式表示的新型N-酰基酸性氨基酸二酰胺衍生物或其盐:其中R 1,R 2,R 3和R 4可以相同或不同,各自表示氢原子取代或未取代的烷基,环烷基,烯基或芳烷基,或R 1和R 2和/或R 3和R 4与各自相邻的氮原子一起形成取代或未取代的杂环基;或R5代表取代或未取代的环烷基,酰基或杂环基; A表示键或取代或未取代的亚烷基,亚烯基或亚链二烯基; n为1、2或3。所述化合物具有对人和动物有效的抗溃疡活性。本公开涉及这种化合物,其制备方法以及包含该化合物的抗溃疡剂。

著录项

  • 公开/公告号ES548221A0

    专利类型

  • 公开/公告日1986-12-16

    原文格式PDF

  • 申请/专利权人 TOYAMA CHEMICAL CO.LTD.;

    申请/专利号ES19850548221

  • 发明设计人

    申请日1985-10-25

  • 分类号C07C103/50;A61K31/16;

  • 国家 ES

  • 入库时间 2022-08-22 07:17:23

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号