首页> 外国专利> ANTICONVULSANT DERIVATIVES USEFUL IN TREATING ALCOANTICONVULSANT DERIVATIVES USEFUL IN TREATING ALCOHOL DEPENDENCY, ADDICTION AND ABUSE HOL DEPENDENCY, ADDICTION AND ABUSE

ANTICONVULSANT DERIVATIVES USEFUL IN TREATING ALCOANTICONVULSANT DERIVATIVES USEFUL IN TREATING ALCOHOL DEPENDENCY, ADDICTION AND ABUSE HOL DEPENDENCY, ADDICTION AND ABUSE

机译:用于治疗酒精依赖,成瘾和滥用的抗惊厥衍生物酒精依赖,成瘾和滥用的抗惊厥衍生物

摘要

A method for treating alcohol dependency, addition and abuse comprising administering to a mammal afflicted with such condition a therapeutically effective amount for treating such condition of a compound of formula (I): wherein X is CH2 or oxygen; R1 is hydrogen or alkyl; and R2, R3, R4 and R5 a re independently hydrogen or lower alkyl and, when X is CH2, R4 and R5 may be alkene groups joined to form a benzene ring and, when X is oxygen, R2 and R3 and/or R4 and R5 together may be a methylenedioxy group of the following formula (II): wherein R6 and R7 are the same or different and are hydrogen, lower alkyl or are alkyl and are joined to form a cyclopentyl or cyclohexyl ring.
机译:一种治疗酒精依赖,加成和滥用的方法,该方法包括对患有这种病症的哺乳动物施用治疗有效量的用于治疗这种病症的式(I)化合物:其中X为CH 2或氧; R1是氢或烷基; R 2,R 3,R 4和R 5分别独立地为氢或低级烷基,并且当X为CH 2时,R 4和R 5可以为连接形成苯环的烯基,并且当X为氧时,R 2和R 3和/或R 4和R5一起可以是下式(II)的亚甲基二氧基:其中R6和R7相同或不同,并且是氢,低级烷基或烷基,并且连接形成环戊基或环己基环。

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