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LAMINATES CONTAINING AN ACTIVE SUBSTANCE FOR TRANSDERMAL SYSTEMS

机译:含有效物质的跨膜系统层压板

摘要

The transdermal system includes a sex hormone-containing adhesive matrix, which contains inclusions of a sex hormone in a hydrophilic non-crosslinked polymer in dissolved or dispersed form. The inclusions have a concentration of 20 to 90 percent by weight of the sex hormone, which is more than 50 percent by weight amorphous. The hydrophilic non-crosslinked polymer can be polyvinylpyrrolidone, methylcellulose, ethylcellulose or hydroxyethylcellulose. The adhesive matrix can be a polyisobutylene, ethylene-vinyl-acetate copolymer or a polystyrene-butadiene block copolymer.
机译:透皮系统包括含性激素的粘合剂基质,该基质含有溶解或分散形式的亲水性非交联聚合物中的性激素包裹体。内含物的浓度为性激素的20-90%(重量),超过50%(重量)的无定形。亲水性非交联聚合物可以是聚乙烯吡咯烷酮,甲基纤维素,乙基纤维素或羟乙基纤维素。粘合剂基质可以是聚异丁烯,乙烯-乙酸乙烯酯共聚物或聚苯乙烯-丁二烯嵌段共聚物。

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