首页> 外国专利> Compounds 6, 7 - deazapurinas N - substituted for Adenosine receptors A1 and A3, a preparation method thereof, a soluble prodrug, Pharmaceutical Composition and Uses Thereof for the manufacture of Medicines and a method for inhibiting the activity of an Adenosine A1 receptor

Compounds 6, 7 - deazapurinas N - substituted for Adenosine receptors A1 and A3, a preparation method thereof, a soluble prodrug, Pharmaceutical Composition and Uses Thereof for the manufacture of Medicines and a method for inhibiting the activity of an Adenosine A1 receptor

机译:取代腺苷受体A1和A3的化合物6、7-脱氮apurinas N,其制备方法,可溶性前药,药物组合物及其在药物生产中的用途以及抑制腺苷A1受体活性的方法

摘要

Compound 7 - 6 deazapurinas N - substituted 1, which has the structure where R3 is a Aromatic Ring of 5-6 members; where R5 and R6 are independently H or alkyl; a method for preparing a water-soluble prodrug, Pharmaceutical Composition and Uses Thereof for Manufacturing d And medicines and a method to inhibit the activity of an a1 adenosine receptor.
机译:化合物7-6的氮杂氮杂嘌呤N-取代的1,具有以下结构:其中R3为5-6元的芳环;其中R5和R6独立地是H或烷基;制备水溶性前药的方法,药物组合物及其在制造药物中的用途和抑制a1腺苷受体活性的方法。

著录项

  • 公开/公告号AR034111A1

    专利类型

  • 公开/公告日2004-02-04

    原文格式PDF

  • 申请/专利权人 OSI PHARMACEUTICALS INC.;

    申请/专利号AR2000P106379

  • 发明设计人

    申请日2000-12-01

  • 分类号C07D487/04;A61K31/519;A61P7/00;A61P7/10;A61P7/12;A61P9/00;A61P9/02;A61P9/04;A61P9/06;A61P9/10;A61P9/12;A61P11/00;A61P11/08;A61P25/00;A61P25/28;

  • 国家 AR

  • 入库时间 2022-08-21 23:12:25

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