首页> 外国专利> COMPLEXES OF E-2-METHOXY-N-(3-{4-3-METHYL-4-(6-METHYL-PYRIDIN-3-YLOXY)-PHENYLAMINO-QUINAZOLIN-6-YL}-ALLYL)-ACETAMIDE, THEIR METHOD OF PRODUCTION, AND USE

COMPLEXES OF E-2-METHOXY-N-(3-{4-3-METHYL-4-(6-METHYL-PYRIDIN-3-YLOXY)-PHENYLAMINO-QUINAZOLIN-6-YL}-ALLYL)-ACETAMIDE, THEIR METHOD OF PRODUCTION, AND USE

机译:E-2-甲氧基-N-(3- {4- [3-甲基-4-(6-甲基-吡啶基-3-羟基)-苯胺基]-喹唑啉-6-基}-烯丙基)-乙酰胺的络合物,他们的生产方法和使用

摘要

The invention relates to complexes of E-2-Methoxy-N-(3-{4-[3-methyl-4-(6-methyl­pyridin-3-yloxy)-phenylamino]-quinazolin-6-yl}-allyl)-acetamide having the following formula I: The invention also relates to pharmaceutical compositions containing the complexes of formula I. The invention further relates to methods of treating hyperproliferative diseases, such as cancers, in mammals, especially humans by administering the above complexes and to methods of preparing the above complexes.
机译:本发明涉及E-2-甲氧基-N-(3- {4- [3-甲基-4-(6-甲基吡啶-3-基氧基)-苯基氨基]-喹唑啉-6-基}-烯丙基)-的配合物。具有下式I的乙酰胺:本发明还涉及含有式I的复合物的药物组合物。本发明还涉及通过施用上述复合物在哺乳动物特别是人中治疗过度增殖性疾病,例如癌症的方法,以及准备上述配合物。

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