首页> 外国专利> Crystalline forms of (1R,2S)-N-(1,1-dimethylethoxy)carbonyl-3-methyl-L-valyl-(4R)-4-(6-methoxy-1-isoquinolinyl)oxy-L-prolyl-1-amino-N-(cyclopropylsulfonyl)-2-ethenyl-cyclopropanecarboxamide, monopotassium salt

Crystalline forms of (1R,2S)-N-(1,1-dimethylethoxy)carbonyl-3-methyl-L-valyl-(4R)-4-(6-methoxy-1-isoquinolinyl)oxy-L-prolyl-1-amino-N-(cyclopropylsulfonyl)-2-ethenyl-cyclopropanecarboxamide, monopotassium salt

机译:(1R,2S)-N-[(1,1-二甲基乙氧基)羰基] -3-甲基-L-戊基-(4R)-4-[(6-甲氧基-1-异喹啉基)氧基] -L的晶体形式-脯氨酰基-1-氨基-N-(环丙基磺酰基)-2-乙烯基-环丙烷甲酰胺,单钾盐

摘要

The present disclosure generally relates to crystalline forms of (1R,2S)-N-[(1,1 -dimethylethoxy)carbonyl]-3-methyl-L-valyl-(4R)-4-[(6-methoxy-1-isoquinolinyl)oxy]-L-prolyl-1-amino-N-(cyclopropylsulfonyl)-2-ethenyl-cyclopropanecarboxamide. The present disclosure also generally relates to a pharmaceutical composition comprising a crystalline form, as well of methods of using a crystalline form in the treatment of Hepatitis C and methods for obtaining such crystalline form.
机译:本公开总体上涉及(1R,2S)-N-[(1,1-二甲基乙氧基)羰基] -3-甲基-L-戊基-(4R)-4-[(6-甲氧基-1-异喹啉基氧基] -L-脯氨酰基-1-氨基-N-(环丙基磺酰基)-2-乙烯基-环丙烷甲酰胺。本公开一般还涉及包含晶型的药物组合物,以及在治疗丙型肝炎中使用晶型的方法以及获得这种晶型的方法。

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