首页> 外国专利> PROCESS FOR THE PREPARATION OF (1S, 4S) - 4 - (3,4 - DICHLOROPHENYL) - 1,2,3,4 -TETRAHYDRO - N - METHYL- 1- NAPHTHYLAMIME HYDROCHLORIDE

PROCESS FOR THE PREPARATION OF (1S, 4S) - 4 - (3,4 - DICHLOROPHENYL) - 1,2,3,4 -TETRAHYDRO - N - METHYL- 1- NAPHTHYLAMIME HYDROCHLORIDE

机译:制备(1S,4S)-4-(3,4-二氯苯酚)-1,2,3,4-四氢-N-甲基-1-萘基氢溴酸盐的过程

摘要

A process for the preparation of (IS,4S)-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-N-methyl-1-naphthylamine hydrochloride, compound of formula I, as crystalline form I or form V directly from compound of formula II or by treating the free base of compound of formula II with amine hydrochloride salt in suitable solvent(s).
机译:制备(IS,4S)-4-(3,4-二氯苯基)-1,2,3,4-四氢-N-甲基-1-萘胺盐酸盐的I型化合物的方法或直接由式II化合物形成V或通过在合适的溶剂中用胺盐酸盐处理式II化合物的游离碱。

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