DERIVATIVES OF 4,6-DIMETHYL-2,3-DIHYDRO-1H-PYRAZOLO4,3-c PYRIDINE-3-ONES AND ETHERS 2,6-DIMETHYL-4-PHENYL-HYDRAZINE NICOTINIC ACIDS AS INTERMEDIATE PRODUCTS FOR THEIR SYNTHESIS, POSSESSING ANTIDEPRESSANT AND ANXIOLYTIC POTENCY

摘要

FIELD: medicine.;SUBSTANCE: invention refers to compounds having anxiolytic and antidepressant activity, which are derivatives of the formula 1 (a-b), or formula 2 (a-b) at that compounds of formula 2 (a-b) are intermediate products in synthesis of compounds of the formula , where R-Cl is a compound 1a or R'=COOC₂H₅ - compound 1b, , where R=COOC₂H₅ and R'=C1 - compound 2a; R=R-COOC₂H₅ - compound 2b.;EFFECT: obtaining new biologically active compounds that differ from analogues as intended in low toxicity and lack of side effects.;5 cl, 3 ex, 5 tbl