首页> 外国专利> NOVEL PROCESS FOR THE PREPARATION OF (2S)-N-((S)-1-((S)-4-METHYL-1-((R)-2- METHYLOXIRAN-2-YL)-1-OXOPENTAN-2-YLCARBAMOYL)-2-PHENYLETHYL)-2-((S)-2-(2- MORPHOLINOACETAMIDO)-4-PHENYLBUTANAMIDO)-4-METHYLPENTANAMIDE

NOVEL PROCESS FOR THE PREPARATION OF (2S)-N-((S)-1-((S)-4-METHYL-1-((R)-2- METHYLOXIRAN-2-YL)-1-OXOPENTAN-2-YLCARBAMOYL)-2-PHENYLETHYL)-2-((S)-2-(2- MORPHOLINOACETAMIDO)-4-PHENYLBUTANAMIDO)-4-METHYLPENTANAMIDE

机译:制备(2S)-N-((S)-1-((S)-4-甲基-1-((R)-2-甲基氧杂环丁-2-基)-1-氧戊烷-2-]的新方法YLCARBAMOYL)-2-PHENYLETHYL)-2-((S)-2-(2-Morpholinoacetamido)-4-PhenylBUTANAMIDO)-4-methentpentanamide

摘要

The present invention relates to novel process for the preparation of (2S)-N-((S)-l-((S)-4-methyl-1 -((R)-2-methyloxiran-2-yl)-1 - oxopentan-2-ylcarbamoyl)-2-phenylethyl)-2-((S)-2-(2-morpholinoacetamido)-4-phenylbutanamido)-4-methylpentanamide represented by the following structural formula-1.
机译:本发明涉及制备(2S)-N-((S)-1-((S)-4-甲基-1-((R)-2-甲基环氧乙烷-2-基)-1)的新方法-由以下结构式-1表示的-氧opentan-2-基氨基甲酰基)-2-苯乙基)-2-((S)-2-(2-吗啉代乙酰胺基)-4-苯基丁酰胺基)-4-甲基戊酰胺。

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