首页> 外国专利> (PIPERIDIN-3-YL)(NAPHTHALEN-2-YL)METHANONE DERIVATIVES AND RELATED COMPOUNDS AS INHIBITORS OF THE HISTONE DEMETHYLASE KDM2B FOR THE TREATMENT OF CANCER

(PIPERIDIN-3-YL)(NAPHTHALEN-2-YL)METHANONE DERIVATIVES AND RELATED COMPOUNDS AS INHIBITORS OF THE HISTONE DEMETHYLASE KDM2B FOR THE TREATMENT OF CANCER

机译:作为组蛋白去甲基化酶KDM2B抑制剂的(哌啶丁-3-基)(萘基-2-基)甲酮衍生物和相关化合物

摘要

The present invention relates to compounds useful as inhibitors of one or more histone demethylses, such as KDM2b. The invention also provides pharmaceutically acceptable compositions comprising compounds of the present invention and methods of using said compositions in the treatment of various disorders.
机译:本发明涉及用作一种或多种组蛋白脱甲基酶的抑制剂的化合物,例如KDM2b。本发明还提供了包含本发明化合物的药学上可接受的组合物,以及使用所述组合物治疗各种疾病的方法。

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