首页> 外国专利> PI 4-KINASE INHIBITOR AS A THERAPEUTIC FOR VIRAL HEPATITIS, CANCER, MALARIA. AUTOIMMUNE DISORDERS AND INFLAMMATION, AND A RADIOSENSITIZER AND IMMUNOSUPPRESSANT

PI 4-KINASE INHIBITOR AS A THERAPEUTIC FOR VIRAL HEPATITIS, CANCER, MALARIA. AUTOIMMUNE DISORDERS AND INFLAMMATION, AND A RADIOSENSITIZER AND IMMUNOSUPPRESSANT

机译:PI 4激酶抑制剂,用于治疗肝炎,疟疾,疟疾。自身免疫疾病和炎症,以及放射增敏剂和免疫抑制剂

摘要

The present invention provides a plant-based flavonoid pharmaceutical composition and its synthetic for inhibition of phosphau'dylinositol-4-kinases and consequent prevention and treatment of RNA viruses including but not limited to viral hepatitis, as well as activity against cancer, malaria, autoimmune disorders and inflammation, prevent organ transplant rejection and as a radiation sensitizer. A method for isolating specific plant-based flavonoid pharmaceutical compositions from raw plant material as well as a method for synthesizing the compositions are also disclosed.
机译:本发明提供了基于植物的类黄酮药物组合物及其合成,其用于抑制磷酸化肌醇-4-激酶并因此预防和治疗RNA病毒,包括但不限于病毒性肝炎,以及针对癌症,疟疾,自身免疫的活性。疾病和炎症,防止器官移植排斥并用作放射增敏剂。还公开了从植物原料中分离特定的基于植物的类黄酮药物组合物的方法以及用于合成该组合物的方法。

著录项

  • 公开/公告号WO2018022868A1

    专利类型

  • 公开/公告日2018-02-01

    原文格式PDF

  • 申请/专利权人 LOWE HENRY C.;TOYANG NGEH J.;

    申请/专利号WO2017US44153

  • 发明设计人 LOWE HENRY C.;TOYANG NGEH J.;

    申请日2017-07-27

  • 分类号A61P31/12;A61K31/33;A61K31/353;C07D311;C07D311/22;C07D311/32;

  • 国家 WO

  • 入库时间 2022-08-21 12:46:04

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