首页> 外国专利> NOVEL SALT OF (R)-(1-METHYLPYRROLIDINE-3-YL)METHYL(3'-CHLORO-4'-FLUORO-1,1'-BIPHENYL-2-YL)CARBAMATE AND A CRYSTAL FORM THEREOF

NOVEL SALT OF (R)-(1-METHYLPYRROLIDINE-3-YL)METHYL(3'-CHLORO-4'-FLUORO-1,1'-BIPHENYL-2-YL)CARBAMATE AND A CRYSTAL FORM THEREOF

机译:(R)-(1-甲基吡咯烷-3-基)甲基(3'-氯-4'-氟-[1,1'-联苯基] -2-基)氨基甲酸酯的新盐及其结晶形式

摘要

NOVEL SALT OF (R)-(1-METHYLPYRROLIDINE-3-YL)METHYL(3'-CHLORO-4'- FLUORO-[1,1'-BIPHENYL]-2-YL)CARBAMATE AND A CRYSTAL FORM THEREOF The present invention relates to a novel salt of (R )-(1-methylpyrrolidine-3- yl)methyl(3'-chloro-4'-fluoro-[1,1'-biphenyl]-2-yl) carbamate and a crystal form thereof. Also, the novel salt of (R)-(1-methylpyrro lidine-3-yl)methyl(3'-chloro-4'- fluoro-[1,1'-biphenyl]-2-yl)carbamate and the cryst al form thereof according to examples of the present invention have remarkably e xcellent stability, hygroscopicity and solubility. [Figure 1]
机译:(R)-(1-甲基吡咯烷-3-基)甲基(3'-氯-4'-氟-[1,1'-联苯基] -2-基)氨基甲酸酯的新盐及其结晶形式本发明涉及一种新型的(R)-(1-甲基吡咯烷-3-基)甲基(3'-氯-4'-氟-[1,1'-联苯] -2-基)氨基甲酸酯的盐及其晶型。另外,(R)-(1-甲基吡咯烷-3-基)甲基(3'-氯-4'-氟-[1,1'-联苯] -2-基)氨基甲酸酯的新颖盐和最根据本发明实施例的其形式具有显着的优异的稳定性,吸湿性和溶解性。 [图1]

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