机译:作为完全拮抗剂的双环核心雌激素:基于桥接氧双环核心芳基磺酰胺的雌激素受体配体的合成,生物学评估和构效关系
Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, Wuhan University School of Pharmaceutical Sciences, Wuhan, 430072, China;
Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, Wuhan University School of Pharmaceutical Sciences, Wuhan, 430072, China;
Department of Cancer Biology, The Scripps Research Institute-Florida,130 Scripps Way, Jupiter, FL 33458, USA;
Department of Cancer Biology, The Scripps Research Institute-Florida,130 Scripps Way, Jupiter, FL 33458, USA;
Department of Cancer Biology, The Scripps Research Institute-Florida,130 Scripps Way, Jupiter, FL 33458, USA;
Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, Wuhan University School of Pharmaceutical Sciences, Wuhan, 430072, China;
Department of Chemistry, University of Illinois, 600 South Mathews Avenue, Urbana, IL 61801, USA;
Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, Wuhan University School of Pharmaceutical Sciences, Wuhan, 430072, China;
Department of Chemistry, University of Illinois, 600 South Mathews Avenue, Urbana, IL 61801, USA;
Department of Cancer Biology, The Scripps Research Institute-Florida,130 Scripps Way, Jupiter, FL 33458, USA;
Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, Wuhan University School of Pharmaceutical Sciences, Wuhan, 430072, China;
机译:含二芳基乙烯基的桥接氧双环核的雌激素受体配体的合成和评价:结构异常的雌激素拮抗剂
机译:含1,1-二芳基乙烯基的桥接双环核是雌激素受体的高亲和力亚型选择性配体。
机译:核受体配体的有希望的核心结构:基于二苯胺骨架的新型雌激素受体配体的设计和合成。
机译:基于药效团的进化方法筛选雌激素受体拮抗剂
机译:设计和合成用于开发亚型选择性雌激素受体配体的新型核心支架。
机译:双环核雌激素为完全拮抗剂:合成雌激素受体的生物学评价并构效关系配位体基于桥接oxabicyclic核心芳基磺酰胺
机译:双环核心雌激素作为完整拮抗剂:基于桥接的长矛核芳基磺酰胺的雌激素受体配体的合成,生物学评价和结构 - 活性关系
机译:LUmI-CELL(商品名)ER(BG1Luc ER Ta)测试方法:用于鉴定人类雌激素受体激动剂和化学品拮抗剂活性的体外测定。 ICCVam测试方法评估报告。