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seen framstella new 6,7 - bensomorfanderivat
seen framstella new 6,7 - bensomorfanderivat
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机译:看到新的弗雷姆斯特拉6,7-贝索莫凡德利瓦
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摘要
The invention is concerned with certain novel 6,7-benzomorphan derivatives having analgesic and/or morphine-antagonistic properties of the formula IMAGE wherein each R is a lower alkyl group; R1 is a hydrogen atom, or an alkyl, haloalkyl, alkenyl, haloalkenyl, alkinyl, cycloalkyl, cycloalkenyl, cycloalkylalkyl, cycloalkenylalkyl, cycloalkylidenealkyl, aralkyl, heteroarylalkyl or heterocycloalkylalkyl group; R2 is a hydrogen atom or a hydroxy, alkoxy, alkoxyalkoxy or acyloxy group.
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机译:本发明涉及某些具有式的镇痛和/或吗啡拮抗特性的新颖的6,7-苯并吗啡衍生物,其中每个R为低级烷基; R1为氢原子,或为烷基,卤代烷基,烯基,卤代烯基,炔基,环烷基,环烯基,环烷基烷基,环烯基烷基,环亚烷基烷基,芳烷基,杂芳基烷基或杂环烷基烷基; R 2是氢原子或羟基,烷氧基,烷氧基烷氧基或酰氧基。
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