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STEROID HORMONE RECEPTOR-SPECIFIC LIGANDS USEFUL FOR TARGETED THERAPY OR MEDICAL IMAGING, IN PARTICULAR CANCER
STEROID HORMONE RECEPTOR-SPECIFIC LIGANDS USEFUL FOR TARGETED THERAPY OR MEDICAL IMAGING, IN PARTICULAR CANCER
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机译:适用于特定癌症的靶向治疗或医学影像的类固醇激素受体配体
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摘要
THE INVENTION CONCERNS LIGANDS SPECIFIC OF STEROID HORMONE RECEPTORS USEFUL FOR TARGETED THERAPY OR IMAGING IN PARTICULAR CANCER HAVING A BASIC STRUCTURAL SKELETON HAVING FOR FORMULA BR/ (CF DRAWING IN BOPI) BR/ According to the invention, they have in particular a hydrophilic or ketone function in position C, a function of chloromethyl in SS on the position C, P / P C A VINYL OR METHYL FUNCTION IN A ON POSITION C AND, / P P D A SUBSTITUTED RADIOACTIVE IODE ON AN ALKYL OR ALKENYL GROUP ATTACHED TO SKELETON, IN PARTICULAR METHYL OR VINYL. / P
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机译:根据本发明,本发明涉及特定的甾族激素受体的特定用途,所述甾族激素受体用于在具有基本结构骨架的特定癌症中用于靶向治疗或成像的特殊癌症。在位置C上具有亲水或酮功能,在位置C上SS中具有氯甲基的功能,C P CA在位置C上具有乙烯基或甲基功能,并且 P>