首页> 外国专利> PIPERIDINE CARBOXYLIC ACID DERIVATIVES AS ROTAMASE ENZYME ACTIVITY INHIBITORS AND USE OF THEM FOR PRODUCING PHARMACEUTICAL COMPOSITIONS SUITABLE FOR TREATING NEUROLOGICAL ACTIVITY

PIPERIDINE CARBOXYLIC ACID DERIVATIVES AS ROTAMASE ENZYME ACTIVITY INHIBITORS AND USE OF THEM FOR PRODUCING PHARMACEUTICAL COMPOSITIONS SUITABLE FOR TREATING NEUROLOGICAL ACTIVITY

机译:哌啶羧酸衍生物作为旋转酶活性抑制剂,并用于生产适于治疗神经活性的药物组合物

摘要

This invention relates to the method of using specially formulated neurotrophic pipecolic acid derivative compounds having an affinity for FKBP-type immunophilins as inhibitors of the enzyme activity associated with immunophilin proteins, and particularly inhibitors of peptidyl-prolyl isomerase or rotamase enzyme activity to stimulate or promote neuronal growth or regeneration.
机译:本发明涉及使用对FKBP型亲免蛋白具​​有亲和力的特殊配制的神经营养性哌酸衍生物化合物作为与亲免蛋白相关的酶活性的抑制剂,特别是肽基-脯氨酰异构酶或旋转酶活性的抑制剂来刺激或促进的方法。神经元生长或再生。

著录项

  • 公开/公告号HU9901752A3

    专利类型

  • 公开/公告日2001-04-28

    原文格式PDF

  • 申请/专利号HU19990001752

  • 发明设计人

    申请日1996-08-26

  • 分类号A61K31/445;

  • 国家 HU

  • 入库时间 2022-08-22 01:25:09

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