首页> 外国专利> 2. Using acid S - (R *, R *) - hexahydro-6 - (2-mercato-1-oxo-3-phenylpropyl) amine-2, 2-dimethyl-7-oxo-1h-azepin-1-acetic as an inhibitor of vasoptimidas to treat isolated earthquake induced hypertension

2. Using acid S - (R *, R *) - hexahydro-6 - (2-mercato-1-oxo-3-phenylpropyl) amine-2, 2-dimethyl-7-oxo-1h-azepin-1-acetic as an inhibitor of vasoptimidas to treat isolated earthquake induced hypertension

机译:2.使用酸[S-(R *,R *)-六氢-6-[(2-巯基-1-氧代-3-苯基丙基)胺-2,2-二甲基-7-氧代-1h-氮杂-1 -乙酸作为血管生成抑制剂的抑制剂,用于治疗孤立的地震诱发的高血压

摘要

It refers to a pharmacological component, including: (a) an acid such as [4S - [4O (R *), 7O, 10a] - octahydro-4 - [(2-mercato-1-oxo-3-phenylpropyl) amino] - 5-oxo-7h-pirido [2, 1-B] [1, 3] tiazepin-7-carboxilico de forma (omaparilat),EL ACIDO S- (RR) -HEXAHIDRO-6- (2-MERCAPTO-1-OXO-3-FENILPROPIL) AMINO-2 2-DIMETIL-7-OXO-1H-AZEPIN-1-ACETICO DE FORMULA II (GEMOPATRILAT) Y vi) INHIBITOR OF THE PLATELET AGGREGATION AS CLOPIDOGREL BISULPHATE, TICLOPIDINE CHLORHYDRATE, ASPIRIN. THE COMPOSITION IS USEFUL TO REDUCE THE FREQUENCY OF CORONARY DISEASE AND THE TREATMENT OF ISOLATED SYSTOLIC HYPERTENSION
机译:它是指药理成分,包括:(a)酸,例如[4S-[4O(R *),7O,10a]-八氢-4-[(2-巯基-1-氧代-3-苯基丙基)氨基]-5-oxo-7h-pirido [2,1-B] [1,3] tiazepin-7-羧甲甲醛(omaparilat),EL ACIDO S-(RR)-HEXAHIDRO-6-(2-MERCAPTO-1 -OXO-3-FENILPROPIL)氨基2 2-二甲基-7-OXO-1H-AZEPIN-1-ACETICO式II(GEMOPATRILAT)Y vi)血小板凝集的抑制剂,如磷脂酰胆碱,硫酸盐,盐酸环氯丁啶,阿司匹林。该组合物可降低冠状动脉疾病的发生率和孤立的系统性高血压的治疗

著录项

  • 公开/公告号PE20011316A1

    专利类型

  • 公开/公告日2002-01-13

    原文格式PDF

  • 申请/专利权人 BRISTOL-MYERS SQUIBB COMPANY;

    申请/专利号PE20060200100

  • 发明设计人 WOLF ROBERT A.;REEVES RICHARD A.;

    申请日2001-04-03

  • 分类号A61K31/00;

  • 国家 PE

  • 入库时间 2022-08-22 00:43:57

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