首页> 外国专利> FIVE-MEMBERED HETEROAROMATIC OLEFINIC AZACYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NCOTINIC CHOLINERGIC RECEPTORS

FIVE-MEMBERED HETEROAROMATIC OLEFINIC AZACYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NCOTINIC CHOLINERGIC RECEPTORS

机译:五元杂芳烃链状氮杂化合物,包含它们的药物组合物及其用作抑制胆碱受体的药物

摘要

The present invention relates to five-membered heteroaromatic olefinic azacyclic compounds and five-membered heteroaromatic acetylenic azacylic compounds, having formula (I) wherein the ring including X, XI, XII, XIII and X IV is heteroaromatic, B is a two-carbon bridging species and Q, E, EI, EII, EIII, m and n are as defined herein and pharmaceutical compositions containing them that are capable of affecting nicotic cholinergic receptors.
机译:具有式(I)的五元杂芳族烯烃氮杂环化合物和五元杂芳族炔属氮杂化合物本发明涉及式(I),其中包括X,XI,XII,XIII和X IV的环为杂芳族,B为二碳桥连种类和Q,E,EI,EII,EIII,m和n如本文所定义,并且包含它们的药物组合物能够影响尼克性胆碱能受体。

著录项

  • 公开/公告号WO2004009599A1

    专利类型

  • 公开/公告日2004-01-29

    原文格式PDF

  • 申请/专利权人 TARGACEPT INC.;CLARK THOMAS JEFFREY;

    申请/专利号WO2002US22997

  • 发明设计人 CLARK THOMAS JEFFREY;

    申请日2002-07-19

  • 分类号C07D487/04;C07D471/04;A61K31/40;A61P25/28;

  • 国家 WO

  • 入库时间 2022-08-21 22:58:47

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