首页> 外国专利> derivatives of n - (arylsulfonyl) beta amino acids containing a substituted group aminomethyle, preparation process and pharmaceutical compositions containing them.

derivatives of n - (arylsulfonyl) beta amino acids containing a substituted group aminomethyle, preparation process and pharmaceutical compositions containing them.

机译:含有取代的氨基甲基的n-(芳基磺酰基)β氨基酸的衍生物,制备方法和含有它们的药物组合物。

摘要

the invention relates to compounds of formula (i): these compounds have a affinite for receivers with a selectivite bradykinin receptors, b1, and can be used for the preparation of medicaments for use in the treatment or prevention of diseases of the will ammation and persistent or chronic inflammatory diseases.
机译:本发明涉及式(i)的化合物:这些化合物对具有选择性的缓激肽受体b1的受体具有一定的亲和力,并且可以用于制备用于治疗或预防遗嘱和持久性疾病的药物。或慢性炎症性疾病。

著录项

  • 公开/公告号TNSN03058A1

    专利类型

  • 公开/公告日2005-04-09

    原文格式PDF

  • 申请/专利权人 SANOFI-SYNTHELABO;

    申请/专利号TN2003SN00058

  • 申请日2002-03-27

  • 分类号C07D295/18;A61K31/198;A61K31/341;A61K31/357;A61K31/36;A61K31/381;A61K31/40;A61K31/4025;A61K31/403;A61K31/417;A61K31/4184;A61K31/422;A61K31/4245;A61K31/426;A61K31/428;A61K31/433;A61K31/435;A61K31/4406;A61K31/4409;A61K31/443;A61K31/445;A61K31/4525;A61K31/454;A61K31/4545;A61K31/4709;A61K31/4725;A61K31/496;A61K31/5377;A61K31/541;A61K31/55;A61P1/00;A61P1/02;A61P1/04;A61P1/16;A61P1/18;A61P3/10;A61P7/00;A61P7/10;A61P9/04;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/00;A61P13/10;A61P13/12;A61P15/00;A61P17/02;A61P17/04;A61P17/06;A61P17/14;A61P19/02;A61P21/00;A61P21/02;A61P25/00;A61P25/04;A61P25/06;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P37/08;A61P43/00;C07C237/30;C07C303/40;C07C311/19;C07D205/04;C07D209/52;C07D211/14;C07D211/16;C07D211/34;C07D211/70;C07D213/40;C07D213/76;C07D215/36;C07D233/54;C07D233/64;C07D271/08;C07D271/12;C07D277/20;C07D277/30;C07D277/80;C07D295/155;C07D295/185;C07D307/52;C07D307/54;C07D307/79;C07D307/81;C07D317/46;C07D317/60;C07D317/66;C07D319/18;C07D333/24;C07D333/62;C07D401/10;C07D405/12;C07D407/12;C07D409/12;C07D409/14;C07D413/12;C07D413/14;C07D417/12;C07D487/08;C07D495/04;

  • 国家 TN

  • 入库时间 2022-08-21 22:16:21

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