首页> 外国专利> derivatives of n - (arylsulfonyl) beta amino acids containing a substituted group aminomethyle, preparation process and pharmaceutical compositions containing them.

derivatives of n - (arylsulfonyl) beta amino acids containing a substituted group aminomethyle, preparation process and pharmaceutical compositions containing them.

机译:含有取代的氨基甲基的n-(芳基磺酰基)β氨基酸的衍生物,制备方法和含有它们的药物组合物。

摘要

the invention relates to compounds of formula (i): these compounds have a affinite for receivers with a selectivite bradykinin receptors, b1, for they can be used.the preparation of medicines intended for the treatment or prevention of disorders of inflammation and persistent or chronic inflammatory diseases.
机译:本发明涉及式(i)的化合物:这些化合物对于具有选择性的缓激肽受体b1的接受者是肯定的,因为它们可以被使用。炎性疾病。

著录项

  • 公开/公告号TNSN03058A1

    专利类型

  • 公开/公告日2005-12-23

    原文格式PDF

  • 申请/专利权人 SANOFI-SYNTHELABO;

    申请/专利号TN2003SN00058

  • 申请日2002-03-27

  • 分类号C07D295/18;A61K31/198;A61K31/341;A61K31/357;A61K31/36;A61K31/381;A61K31/40;A61K31/4025;A61K31/403;A61K31/417;A61K31/4184;A61K31/422;A61K31/4245;A61K31/426;A61K31/428;A61K31/433;A61K31/435;A61K31/4406;A61K31/4409;A61K31/443;A61K31/445;A61K31/4525;A61K31/454;A61K31/4545;A61K31/4709;A61K31/4725;A61K31/496;A61K31/5377;A61K31/541;A61K31/55;A61P1;A61P1/02;A61P1/04;A61P1/16;A61P1/18;A61P3/10;A61P7;A61P7/10;A61P9/04;A61P9/10;A61P11;A61P11/02;A61P11/06;A61P13;A61P13/10;A61P13/12;A61P15;A61P17/02;A61P17/04;A61P17/06;A61P17/14;A61P19/02;A61P21;A61P21/02;A61P25;A61P25/04;A61P25/06;A61P25/28;A61P27/02;A61P27/06;A61P29;A61P37/08;A61P43;C07C237/30;C07C303/40;C07C311/19;C07D205/04;C07D209/52;C07D211/14;C07D211/16;C07D211/34;C07D211/70;C07D213/40;C07D213/76;C07D215/36;C07D233/54;C07D233/64;C07D271/08;C07D271/12;C07D277/20;C07D277/30;C07D277/80;C07D295/155;C07D295/185;C07D307/52;C07D307/54;C07D307/79;C07D307/81;C07D317/46;C07D317/60;C07D317/66;C07D319/18;C07D333/24;C07D333/62;C07D401/10;C07D405/12;C07D407/12;C07D409/12;C07D409/14;C07D413/12;C07D413/14;C07D417/12;C07D487/08;C07D495/04;

  • 国家 TN

  • 入库时间 2022-08-21 21:37:41

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