首页> 外国专利> APPLICATION OF A PYRAZOLE DERIVATIVE FOR THE PRODUCTION OF A MEDICINE SUITABLE FOR PREVENTION AND TREATMENT OF DYSLIPIDEMIA AND DISEASES ASSOCIATED WITH DYSLIPIDEMIA AND / OR OBESITY

APPLICATION OF A PYRAZOLE DERIVATIVE FOR THE PRODUCTION OF A MEDICINE SUITABLE FOR PREVENTION AND TREATMENT OF DYSLIPIDEMIA AND DISEASES ASSOCIATED WITH DYSLIPIDEMIA AND / OR OBESITY

机译:吡唑衍生物在生产适于预防和治疗血脂异常和与血脂异常和/或肥胖有关的疾病的药物中的应用

摘要

Use of a pyrazole compound (I) which is an antagonist of the CB 1 cannabinoid receptor to prepare a composition for treatment and prevention of metabolic syndrome. An independent claim is also included for a composition containing (I) and a second active agent (II). ACTIVITY : Antilipemic; Anorectic; Antidiabetic; Cardiant; Hypotensive; Antiarteriosclerotic; Antianginal; Anticoagulant; Cerebroprotective; Ophthalmological; Hepatotropic. MECHANISM OF ACTION : CB 1 cannabinoid receptor antagonist.
机译:作为CB 1大麻素受体拮抗剂的吡唑化合物(I)在制备用于治疗和预防代谢综合征的组合物中的用途。对于包含(I)和第二活性剂(II)的组合物也包括独立权利要求。活动:抗血脂;厌食的;抗糖尿病卡迪恩降压;抗动脉硬化;抗心绞痛抗凝物;脑保护眼科肝的。作用机理:CB 1大麻素受体拮抗剂。

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