首页> 外国专利> N-(3-ETHYNYLPHEYL)-6,7-BIS(2-METHOXYETHOXY)-4-QUINAZOLINAMINE MESYLATE ANHYDRATE AND MONOHYDRATE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME

N-(3-ETHYNYLPHEYL)-6,7-BIS(2-METHOXYETHOXY)-4-QUINAZOLINAMINE MESYLATE ANHYDRATE AND MONOHYDRATE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME

机译:N-(3-乙炔基)-6,7-双(2-甲氧基乙氧基)-4-喹唑啉磺酸甲酯的甲酸酐,甲酸酯和含有相同成分的药物组合物

摘要

The present invention relates to the anhydrous and hydrate forms of N- (3-ethynylphenyl)-6,7-bis (2-methoxyethoxy)4-quinazolinamine mesylate. The invention also relates to pharmaceutical compositions containing N- (3-ethynylphenyl)-6,7- bis(2-methoxyethoxy) -4-quinazolinamine mesylate and to methods of treating hyperproliferative disorders, such as cancer, by administering N- (3-ethynylphenyl)-6,7- bis(2-methoxyethoxy)-4- quinazolinamine mesylate.
机译:本发明涉及N-(3-乙炔基苯基)-6,7-双(2-甲氧基乙氧基)4-喹唑啉胺甲磺酸盐的无水和水合物形式。本发明还涉及含有N-(3-乙炔基苯基)-6,7-双(2-甲氧基乙氧基)-4-喹唑啉胺甲磺酸盐的药物组合物,以及通过施用N-(3-乙炔基苯基)-6,7-双(2-甲氧基乙氧基)-4-喹唑啉胺甲磺酸盐。

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