首页> 外国专利> BENZOTHIENO 3,2-cPYRAZOLYL AND BENZOFURANO 3,2-c PYRAZOLYL COMPOUNDS, THEIR USE IN DISEASES ASSOCIATED WITH THE 5-HT_2C RECEPTOR AND INTERMEDIATE COMPOUNDS THEREOF

BENZOTHIENO 3,2-cPYRAZOLYL AND BENZOFURANO 3,2-c PYRAZOLYL COMPOUNDS, THEIR USE IN DISEASES ASSOCIATED WITH THE 5-HT_2C RECEPTOR AND INTERMEDIATE COMPOUNDS THEREOF

机译：苯并噻吩并[3,2- c ]吡唑基和苯并呋喃并[3,2- c ]吡唑基化合物，它们与5-HT _{2C相关的疾病中使用/ Sub>受体及其中间化合物}

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Disclosed are benzothieno[3,2-c]pyrazolyl and benzofurano[3,2-c]pyrazolyl compounds of the formula (I) and (II), and intermediates of the formula (Ia) and (IIa) which are tautomers, wherein the variables A, X, y, R¹, R², R³ and R⁴ are as defined in the specification. The compounds are useful for the treatment or prevention of diseases and/or behaviors involving the 5-HT_2C receptor site. 展开▼

机译：公开了式（I）和（II）的苯并噻吩并[3,2- c ]吡唑基和苯并呋喃并[3,2- c ]吡唑基化合物及其中间体为互变异构体的式（Ia）和（IIa），其中变量A，X，y，R ^{1 ，R ^{2 ，R ^{3 和R ^{4 如规范中所定义。这些化合物可用于治疗或预防涉及5-HT _{2C 受体位点的疾病和/或行为。}}}}} 展开▼

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公开/公告号WO03057161A3

专利类型

公开/公告日2011-08-04

原文格式PDF

申请/专利权人 BAYER PHARMACEUTICALS CORPORATION;LADOUCEUR GAETAN H.;CHOI SOONGYOU;WANG YAMIN;
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申请/专利号WO2002US41859

发明设计人 LADOUCEUR GAETAN H.;CHOI SOONGYOU;WANG YAMIN;
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申请日2002-12-28

分类号C07D491/048;C07D495/04;A61K31/4162;A61P3;A61P25;

国家 WO

入库时间 2022-08-21 18:01:06

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