首页> 外国专利> CARVEDILOL PHOSPHATE SALTS OR SOLVATES THEREOF, CORRESPONDING COMPOSITIONS AND USES THEREOF IN THE PREPARATION OF MEDICAMENTS FOR TREATING HYPERTENSION, CONGESTIVE HEART FAILURE OR ANGINA

CARVEDILOL PHOSPHATE SALTS OR SOLVATES THEREOF, CORRESPONDING COMPOSITIONS AND USES THEREOF IN THE PREPARATION OF MEDICAMENTS FOR TREATING HYPERTENSION, CONGESTIVE HEART FAILURE OR ANGINA

机译:卡维地洛磷酸盐或它们的盐,相应的成分以及在制备治疗高血压,充血性心力衰竭或心绞痛的药物中的用途

摘要

The present invention relates to carvedilol phosphate salts, which include novel crystalline forms of carvedilol dihydrogen phosphate (i.e., dihydrogen phosphate salt of 1-(carbazol-4-yloxy-3-[[2-(o-methoxyphenoxy)ethyl]amino]-2-propanol) and/or carvedilol hydrogen phosphate, etc.), and/or solvates thereof, compositions containing the aforementioned salts and/or solvates, and methods of using the aforementioned salts and/or solvates to treat hypertension, congestive heart failure and angina, etc.
机译:本发明涉及卡维地洛磷酸盐,其包括卡维地洛磷酸二氢盐的新结晶形式(即1-(咔唑-4-基氧基-3-[[2-(邻甲氧基苯氧基)乙基]氨基]-磷酸二氢盐)。 2-丙醇和/或卡维地洛磷酸氢盐等)和/或其溶剂化物,包含上述盐和/或溶剂化物的组合物以及使用上述盐和/或溶剂化物治疗高血压,充血性心力衰竭和心绞痛等

著录项

  • 公开/公告号IL165814A

    专利类型

  • 公开/公告日2012-05-31

    原文格式PDF

  • 申请/专利号IL20040165814

  • 发明设计人

    申请日2004-12-16

  • 分类号A61K31/403;A61P9;A61P9/04;A61P9/12;C07D209/82;C07D209/88;

  • 国家 IL

  • 入库时间 2022-08-21 17:24:49

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