首页> 外国专利> PENTAFLUOROSULFANYL BENZOYLGUANIDINES, METHOD FOR THEIR PRODUCTION, THEIR USE AS MEDICAMENTS OR DIAGNOSTIC AGENTS AND MEDICAMENT CONTAINING THE SAME

PENTAFLUOROSULFANYL BENZOYLGUANIDINES, METHOD FOR THEIR PRODUCTION, THEIR USE AS MEDICAMENTS OR DIAGNOSTIC AGENTS AND MEDICAMENT CONTAINING THE SAME

机译:五氟磺酰苯甲酰胍,其生产方法,其用作药物或诊断剂的用途以及包含该成分的药物

摘要

The invention relates to pentafluorosulfanyl benzoylguanidines of formula (I), in which R1 to R4 are defined as cited in the claims. Said substances are suitable for use as anti-arrhythmic medicaments comprising cardio-protective components for the prophylaxis and treatment of infarcts, in addition to the treatment of angina pectoris. They also preventatively inhibit the pathophysiological events that occur during ischaemically induced traumas, in particular during the triggering of ischaemically induced cardiac arrhythmia.
机译:本发明涉及式(I)的五氟硫烷基苯甲酰基胍,其中R 1至R 4如权利要求中所定义。所述物质适合用作抗心律失常药物,其除了治疗心绞痛外还包含用于预防和治疗梗塞的心脏保护性成分。它们还预防性抑制在局部缺血引起的创伤期间发生的病理生理事件,特别是在引起局部缺血引起的心律不齐的过程中。

著录项

  • 公开/公告号IN252114B

    专利类型

  • 公开/公告日2012-05-04

    原文格式PDF

  • 申请/专利权人

    申请/专利号IN1646/CHENP/2006

  • 发明设计人 KLEEMANN HEINZ-WERNER;

    申请日2006-05-11

  • 分类号A61K31/166;C07C381;

  • 国家 IN

  • 入库时间 2022-08-21 17:23:55

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号