首页> 外国专利> SUBSTITUTED (5H-PYRROLO2,1-C1,4BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS

SUBSTITUTED (5H-PYRROLO2,1-C1,4BENZODIAZEPIN-11-YL)PIPERAZIN-1-YL-2,2-DIMETHYLPROPANOIC ACID COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS

机译:替代[(5H-吡咯并[2,1-C] [1,4]苯二氮杂PIN基-11-基)哌嗪-1-基] -2,2-二甲基丙酸化合物作为双重活性H1逆向激动剂/ 5-HT2A拮抗剂

摘要

A dual H1/5-HT2A receptor antagonist of the formula:, its uses, and methods for its preparation are described.
机译:描述了下式的双重H1 / 5-HT2A受体拮抗剂:其用途及其制备方法。

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