首页> 外国专利> COMPOUNDS, PROCESSED FOR THE MANUFACTURE, PHARMACEUTICAL COMPOSITIONS UNDERSTANDING THEM, METHOD FOR TREATMENT AND / OR PREVENTION OF NURSES THAT ARE ASSOCIATED WITH THE MODULATION OF BUBY 5 SST RECEIVERS AND USE OF THESE COMPOUNDS.

COMPOUNDS, PROCESSED FOR THE MANUFACTURE, PHARMACEUTICAL COMPOSITIONS UNDERSTANDING THEM, METHOD FOR TREATMENT AND / OR PREVENTION OF NURSES THAT ARE ASSOCIATED WITH THE MODULATION OF BUBY 5 SST RECEIVERS AND USE OF THESE COMPOUNDS.

机译:用于制造的化合物,理解其的药物组合物,与BUBY 5 SST受体的调节有关的治疗和/或预防营养的方法以及这些化合物的使用。

摘要

This invention relates to 4,4-disubstituted piperidine derivatives of the formula wherein A and R1 to R5 are as defined in the specification, and pharmaceutically acceptable salts thereof. The invention further relates to pharmaceutical compositions containing such compounds, to a process for their preparation and to their use for the treatment and/or prevention of diseases which are associated with the modulation of SST receptors subtype 5.
机译:本发明涉及下式的4,4-二取代哌啶衍生物及其药学上可接受的盐,其中A和R 1至R 5如说明书中所定义。本发明进一步涉及含有此类化合物的药物组合物,其制备方法以及其在治疗和/或预防与SST受体5亚型调节有关的疾病中的用途。

著录项

  • 公开/公告号BRPI0812302A2

    专利类型

  • 公开/公告日2014-11-25

    原文格式PDF

  • 申请/专利权人 F. HOFFMANN-LA ROCHE AG;

    申请/专利号BR2008PI12302

  • 申请日2008-05-15

  • 分类号C07D211/66;A61K31/435;A61K31/4468;A61K31/455;A61P3;C07D401/12;C07D471/10;

  • 国家 BR

  • 入库时间 2022-08-21 15:16:09

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