首页> 外国专利> Crystalline form of d,l- malate hemihydrate salt of (3s,5s)-7-3-amino-5-methyl-piperidinyl-1- cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3- quinoline carboxylic acid and pharmaceutical composition for use for infectious disorders

Crystalline form of d,l- malate hemihydrate salt of (3s,5s)-7-3-amino-5-methyl-piperidinyl-1- cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3- quinoline carboxylic acid and pharmaceutical composition for use for infectious disorders

机译:(3s,5s)-7- [3-氨基5-甲基-哌啶基] -1-环丙基-1,4-二氢-8-甲氧基-4-氧代-3的d,l-苹果酸半水合物盐的晶体形式-用于传染性疾病的喹啉羧酸和药物组合物

摘要

The present invention is directed to malate salts of (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid, and its polymorphs. The present invention is also directed to pharmaceutical compositions comprising the described salts and polymorphs.
机译:本发明涉及(3S,5S)-7- [3-氨基5-甲基-哌啶基] -1-环丙基-1,4-二氢-8-甲氧基-4-氧代-3-喹啉羧酸的苹果酸盐。酸及其多晶型物。本发明还涉及包含所述盐和多晶型物的药物组合物。

著录项

  • 公开/公告号IL193990A

    专利类型

  • 公开/公告日2014-12-31

    原文格式PDF

  • 申请/专利权人 THE PROCTER & GAMBLE COMPANY;

    申请/专利号IL20080193990

  • 发明设计人

    申请日2008-09-09

  • 分类号C07D;

  • 国家 IL

  • 入库时间 2022-08-21 15:15:25

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