首页> 外国专利> ESTROGEN RECEPTOR .BETA. PARTIAL AGONIST HAVING ESTROGEN RECEPTOR .ALPHA. INHIBITORY EFFECT, AND GYNECOLOGICAL DISEASE THERAPEUTIC AGENT USING SAME

ESTROGEN RECEPTOR .BETA. PARTIAL AGONIST HAVING ESTROGEN RECEPTOR .ALPHA. INHIBITORY EFFECT, AND GYNECOLOGICAL DISEASE THERAPEUTIC AGENT USING SAME

机译:雌激素受体。具有雌激素受体.ALPHA的部分激动剂。相同的抑制作用和妇科疾病治疗剂

摘要

[Problem] To provide a therapeutic agent for estrogen-dependent gynecological disorders such as endometriosis, uterine fibroids, and adenomyosis. [Solution] An estrogen receptor a-inhibiting ß partial agonist represented by structural formula (a), a pharmaceutically-acceptable salt thereof, or a hydrate of either of the aforementioned is used as an active ingredient.
机译:[问题]为子宫内膜异位,子宫肌瘤,子宫腺肌病等雌激素依赖性妇科疾病提供治疗剂。 [解决方案]使用由结构式(a)表示的雌激素受体α抑制性β部分激动剂,其药学上可接受的盐或上述任何一种的水合物作为活性成分。

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