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A LIPID NANOPARTICLE FOR CARRYING ANTISENSE OLIGONUCLEOTIDES INHIBITING BCL-2 AND METHOD FOR PREPARING THE SAME
A LIPID NANOPARTICLE FOR CARRYING ANTISENSE OLIGONUCLEOTIDES INHIBITING BCL-2 AND METHOD FOR PREPARING THE SAME
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机译:用于携带抑制BCL-2的反义寡核苷酸的脂质纳米颗粒及其制备方法
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摘要
A lipid nanoparticle for antisense oligonucleotides inhibiting bcl-2 and belonging to the technical field of biology. The lipid nanoparticle for antisense oligonucleotides inhibiting bcl-2 is prepared by coating an antisense oligonucleotide with a membrane material, and the nucleic acid sequence is 5′-TCT CCC AGC GTG CGC CAT-3′ (SEQ ID NO: 1), or 5′ UCU CCC AGC GTG CGC CAU 3′ (SEQ ID NO: 2). And a method for preparing the same is provided. The nanoparticles have a fairly good inhibitory effect on the growth of tumor cells and specific target genes, and particularly have a fairly good inhibitory effect on KB cervical cancer cells.
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机译:用于抑制bcl-2的反义寡核苷酸的脂质纳米颗粒,属于生物学技术领域。通过用膜材料包被反义寡核苷酸来制备用于反义寡核苷酸抑制bcl-2的脂质纳米颗粒,并且核酸序列是5'-TCT CCC AGC GTG CGC CAT-3'(SEQ ID NO:1)或5 'UCU CCC AGC GTG CGC CAU 3'(SEQ ID NO:2)。并提供了一种制备方法。纳米粒子对肿瘤细胞和特定靶基因的生长具有相当好的抑制作用,特别是对KB宫颈癌细胞具有相当好的抑制作用。
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