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Novel compounds having inhibitory activity against sodium-dependant glucose transporter

机译:对钠依赖性葡萄糖转运蛋白具有抑制活性的新型化合物

摘要

A compound of the formula: wherein Ring A and Ring B are: (1) Ring A is an optionally substituted unsaturated monocyclic heterocyclic ring, and Ring B is an optionally substituted unsaturated monocyclic heterocyclic ring, an optionally substituted unsaturated fused heterobicyclic ring, or an optionally substituted benzene ring, (2) Ring A is an optionally substituted benzene ring, and Ring B is an optionally substituted unsaturated monocyclic heterocyclic ring or an optionally substituted unsaturated fused heterobicyclic ring, or (3) Ring A is an optionally substituted unsaturated fused heterobicyclic ring, and Ring B are independently an optionally substituted unsaturated monocyclic heterocyclic ring, an optionally substituted unsaturated fused heterobicyclic ring, or an optionally substituted benzene ring; X is a carbon atom or a nitrogen atom; Y is ۥ(CH 2 ) n -(n is 1 or 2); a pharmaceutically acceptable salt thereof, or a prodrug thereof.
机译:下式的化合物:其中环A和环B为:(1)环A为任选取代的不饱和单环杂环,并且环B为任选取代的不饱和单环杂环,任选取代的不饱和稠合杂环二环或任选取代的苯环,( 2)环A为任选取代的苯环,环B为任选取代的不饱和单环杂环或任选取代的不饱和稠合杂环二环,或(3)环A为任选取代的不饱和稠合杂环二环,且环B为独立地为任选取代的不饱和单环杂环,任选取代的不饱和稠合杂环二环或任选取代的苯环; X是碳原子或氮原子; Y为€•(CH 2)n-(n为1或2);其药学上可接受的盐或其前药。

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