Design and Synthesis of Novel Pyrazolo[3,4-d]pyrimidin-1-yl piperidine Derivatives as Bruton's Tyrosine Kinase Inhibitors

Park Hyebin; Park Chi Hoon; Kang Seung-Tae; Jeon Jeong Hee; Archary Raghavendra; Lee Joo-Youn; Kim Pilho; Jung Heejung; Yun Chang-Soo; Hwang Jong Yeon; Ryu Do Hyun; Cho Sung Yun

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Design and Synthesis of Novel Pyrazolo[3,4-d]pyrimidin-1-yl piperidine Derivatives as Bruton's Tyrosine Kinase Inhibitors

机译：设计和合成新型吡唑啉[3,4-D]嘧啶-1-基哌啶衍生物作为Bruton的酪氨酸激酶抑制剂

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来源
《Bulletin of the Korean Chemical Society》 |2017年第2期|共4页
作者
Park Hyebin; Park Chi Hoon; Kang Seung-Tae; Jeon Jeong Hee; Archary Raghavendra; Lee Joo-Youn; Kim Pilho; Jung Heejung; Yun Chang-Soo; Hwang Jong Yeon; Ryu Do Hyun; Cho Sung Yun;
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作者单位

Sungkyunkwan Univ Dept Chem Suwon 440746 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Sungkyunkwan Univ Dept Chem Suwon 440746 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

Sungkyunkwan Univ Dept Chem Suwon 440746 South Korea;

Korea Res Inst Chem Technol Drug Discovery Div Daejeon 305606 South Korea;

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原文格式 PDF
正文语种 eng
中图分类化学;
关键词
Bruton's tyrosine kinase; BTK inhibitor; Pyrimidine derivative; Kinase inhibitor; Anticancer agent;

机译：Btron的酪氨酸激酶;BTK抑制剂;嘧啶衍生物;激酶抑制剂;抗癌剂;

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Design and Synthesis of Novel Pyrazolo[3,4-d]pyrimidin-1-yl piperidine Derivatives as Bruton's Tyrosine Kinase Inhibitors

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