机译:二孔豆类对九种细胞色素P450同种型,UGTS和三种药物转运蛋白的影响
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
College of Food Science and Technology Shanghai Ocean University;
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
State Key Laboratory of Genetic Engineering Institute of Genetics School of Life Sciences Fudan;
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
Department of Pharmacy Shanghai Jiao Tong University Affiliated Sixth People's Hospital;
Diosmetin; Cytochrome P450; UDP-glucuronyltransferases; Hepatic uptake transporters; Drug-drug interactions;
机译:二孔豆类对九种细胞色素P450同种型,UGTS和三种药物转运蛋白的影响
机译:黄酮类地索美汀和橙皮素是细胞色素P450 2C9介导的体外药物代谢的有效抑制剂。
机译:类黄酮Diosmetin和橙皮素是细胞色素P450 2C9介导的体外药物代谢的有效抑制剂。
机译:菊花素对人细胞色素P450 1A2的同工型选择性抑制。动力学分析,分子对接和分子动力学模拟
机译:饮食对药物代谢和转运的影响:薄荷油,圣约翰草和果汁对体外和人体中细胞色素P450 3A4,P-糖蛋白和有机阴离子转运多肽的影响
机译:UDP-葡糖醛糖基转移酶(UGT)介导的细胞色素P450 3A4活性的衰减:UGT同种型抑制机制
机译:细胞色素P450 3A4改变UDP-葡萄糖醛酸转移酶1A亚家族的功能:UGT亚型和UGT1A1 / 7变体的敏感性不同。