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机译:2-(4-(((2 - (((2 - (((2 - ((2 - ((2 - ((2 - ((2 - ((2 - ((2 - ((2 - )乙基)乙基)哌嗪-1-基)-N-(6-甲基-2, 4-双(甲硫硫胺)吡啶-3-基)乙酰胺盐酸盐[K-604],酰基-CoA:胆固醇O-酰基转移酶-1抑制剂
Kowa Co Ltd Pharmaceut Div Tokyo New Drug Res Labs 2-17-43 Noguchicho Tokyo 1890022 Japan;
Kowa Co Ltd Pharmaceut Div Tokyo New Drug Res Labs 2-17-43 Noguchicho Tokyo 1890022 Japan;
Kowa Co Ltd Pharmaceut Div Tokyo New Drug Res Labs 2-17-43 Noguchicho Tokyo 1890022 Japan;
Kowa Co Ltd Pharmaceut Div Fuji Res Labs 332-1 Ohnoshinden Fuji Shizuoka 4178650 Japan;
Kowa Co Ltd Pharmaceut Div Tokyo New Drug Res Labs 2-17-43 Noguchicho Tokyo 1890022 Japan;
Acyl-CoA:cholesterol O-acyltransferase; ACAT-1 inhibitor; K-604; Metabolite; Monosulfoxidation; Pharmacokinetics; Microsomes; Clearance; CYP3A4; Metabolic pattern;
机译:2-(4-(((2 - (((2 - (((2 - ((2 - ((2 - ((2 - ((2 - ((2 - ((2 - ((2 - )乙基)乙基)哌嗪-1-基)-N-(6-甲基-2, 4-双(甲硫硫胺)吡啶-3-基)乙酰胺盐酸盐[K-604],酰基-CoA:胆固醇O-酰基转移酶-1抑制剂
机译:2-(4-(((2 - (((2 - (((2 - ((2 - ((2 - ((2 - ((2 - ((2 - ((2 - ((2 - )乙基)乙基)哌嗪-1-基)-N-(6-甲基-2, 4-双(甲硫硫胺)吡啶-3-基)乙酰胺盐酸盐[K-604],酰基-CoA:胆固醇O-酰基转移酶-1抑制剂
机译:发现临床候选2-(4-(2 - ((2 - ((1H-苯并[D] Imidazol-2-Y1))乙基)哌嗪-1-基)-N-(6-甲基-2,4-双( 甲硫基)吡啶-3-基)氯胺盐酸盐[K-604],一种水溶性酰基-CoA:胆固醇O-酰基转移酶-1抑制剂
机译:2 - [[5-烷基/芳烷基取代-1,3,4-恶二唑-2-基]硫代] -N- [4-(4-吗啉基)苯基]乙酰胺衍生物的合成,抗菌评价和溶血活性