机译:BMS-986260发现有效,选择性和口服生物利用的TGFβR1抑制剂作为免疫肿瘤剂
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Biocon Bristol Myers Squibb R&
D Ctr Bangalore 560099 KA India;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Rigel Pharmaceut Inc San Francisco CA 94080 USA;
Rigel Pharmaceut Inc San Francisco CA 94080 USA;
Rigel Pharmaceut Inc San Francisco CA 94080 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
Bristol Myers Squibb Res &
Dev Princeton NJ 08543 USA;
TGF beta R1; immuno-oncology; imidazo-pyridine; imidazo-pyridazine; intermittent dosing;
机译:BMS-986260发现有效,选择性和口服生物利用的TGFβR1抑制剂作为免疫肿瘤剂
机译:发现有效,选择性和口服可生物利用的PDE9抑制剂作为潜在的降血糖药。
机译:发现2-((R)-4-(2-氟-4-(甲基磺酰基)苯基)-2-甲基哌嗪-1-基)-N-(((1R,2s,3S,5S,7S)-5-羟基金刚烷-2-y1)嘧啶-4-羧酰胺(SKI2852):一种11型β-羟基类固醇脱氢酶(11 beta-HSD1)的高效,选择性和口服生物利用度抑制剂
机译:CNX-774,Bruton的酪氨酸激酶的不可逆转,选择性和口服生物可利用的抑制剂:体外Adme,选择性和药代动力学性能
机译:寻找选择性和有效的高尔基α-甘露糖苷酶II抑制剂作为潜在的抗癌药:3-取代-swainsonine类似物的合成和在固体支持物上固定的swainsonine类似物的制备。
机译:发现BMS-986260有效选择性和口服生物可利用的TGFβR1抑制剂作为免疫肿瘤学剂
机译:发现GLPG1972 / S201086,有效,选择性和口服生物的ADAMTA-5用于治疗骨关节炎的抑制剂