机译:一种异喹啉脚手架作为一种新型的血糖HIV-1整合酶抑制剂
Division of Medicinal Chemistry &
Pharmacognosy College of Pharmacy The Ohio State University;
Division of Infectious Diseases University of Colorado School of Medicine;
Division of Infectious Diseases University of Colorado School of Medicine;
Division of Infectious Diseases University of Colorado School of Medicine;
Division of Pharmaceutics &
Pharmaceutical Chemistry College of Pharmacy The Ohio State University;
Division of Medicinal Chemistry &
Pharmacognosy College of Pharmacy The Ohio State University;
Division of Medicinal Chemistry &
Pharmacognosy College of Pharmacy The Ohio State University;
Division of Pharmaceutics &
Pharmaceutical Chemistry College of Pharmacy The Ohio State University;
Division of Infectious Diseases University of Colorado School of Medicine;
Division of Medicinal Chemistry &
Pharmacognosy College of Pharmacy The Ohio State University;
allosteric inhibitor; HIV-1 integrase; protein multimerization;
机译:一种异喹啉脚手架作为一种新型的血糖HIV-1整合酶抑制剂
机译:HIV-1复制早期,变构HIV-1整合酶抑制剂BI / D和LEDGF / p75之间的竞争相互作用不利地影响了抑制剂的效力。
机译:开发下一代HIV-1整合酶抑制剂:吡唑酮作为新型抑制剂支架。
机译:使用HDX质谱法对HIV整合酶进行颠覆抑制剂作用机理的特征
机译:机械和结构研究进入颠覆性HIV-1整合酶抑制剂的作用方式
机译:一类新型的变构HIV-1整合酶抑制剂通过催化核心域的晶体学片段筛选确定。
机译:变构HIV-1整合酶抑制剂导致病毒RNA基因组过早降解并整合到靶细胞中