机译:发现2 - [(e)-2-(7-氟-3-甲基喹喔啉-2-基)乙烯基] -6-吡咯烷-1-基-N-(四氢-2H-吡喃-4-基)嘧啶 - 4-氨盐酸盐作为高选择性PDE10A抑制剂
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp 2-2-50 Kawagishi Toda Saitama 3358505 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
Mitsubishi Tanabe Pharma Corp Aoba Ku 1000 Kamoshida Cho Yokohama Kanagawa 2270033 Japan;
phosphodiesterase (PDE) 10A; schizophrenia; conditioned avoidance response (CAR); stilbene; quinoxaline; pyrimidine;
机译:2-[((E)-2-(7-Fluoro-3-methylquinoxalin-2-yl)vinyl] -6-pyrrolidin-1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-的发现4-胺盐酸盐作为高选择性PDE10A抑制剂
机译:N-(2-({2-(((2S)-2-cyanopyrrolidin-1-yl)-2-oxoethyl} amino)-2-methylpropyl)-2-methyl pyrazolo(1,5-a)的发现和药理特性嘧啶-6-羧酰胺盐酸盐(那格列汀盐酸盐)作为有效的选择性DPP-IV抑制剂。
机译:发现(e)-N-1-(3-氟苯基)-N-3-(3-(2-(吡啶-2-基)乙烯基)-1H-吲唑-6-Y1)丙二酰胺(CHMFL-kit- 033)作为胃肠道间质瘤的新型C-kit T670i突变体选择性激酶抑制剂(GISTS)
机译:微波辅助制备2-(苄硫基)咪唑和2-(苄硫基)苯并咪唑及其与2-巯基咪唑和2-巯基苯并咪唑的比较缓蚀性能
机译:合成5- [2-(5-ami基苯并咪唑基)]-2-(4-ami基苯基)呋喃盐酸盐的类似物以测试DNA小沟二聚体结合模型。
机译:两种Cathinone衍生物的光谱和晶体学表征:1-(4-氟苯基)-2-(甲基氨基)戊丹-1-酮盐酸盐(4-FPD)和1-(4-甲基苯基)-2-(乙基氨基)戊丹-1一(4-MEAP)盐酸盐
机译:发现2 - ( e i>) - 2-(7-氟-3-甲基喹喔啉-2-基)乙烯基 -6-Pyrrolidin-1-Y1- N I> - (四氢-2 H氢吡喃-4-基)嘧啶-4-氨基盐酸盐作为高度选择性PDE10A抑制剂