机译:发现(e)-N-1-(3-氟苯基)-N-3-(3-(2-(吡啶-2-基)乙烯基)-1H-吲唑-6-Y1)丙二酰胺(CHMFL-kit- 033)作为胃肠道间质瘤的新型C-kit T670i突变体选择性激酶抑制剂(GISTS)
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Precis Med Res Lab Anhui Prov Hefei 230088 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Precis Med Res Lab Anhui Prov Hefei 230088 Anhui Peoples R China;
Univ Pittsburgh Univ Pittsburgh Canc Inst Dept Radiol Mol Imaging Lab Pittsburgh PA 15219 USA;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
Chinese Acad Sci Hefei Inst Phys Sci Key Lab High Magnet Field &
Ion Beam Phys Biol High Magnet Field Lab Hefei 230031 Anhui Peoples R China;
机译:发现(e)-N-1-(3-氟苯基)-N-3-(3-(2-(吡啶-2-基)乙烯基)-1H-吲唑-6-Y1)丙二酰胺(CHMFL-kit- 033)作为胃肠道间质瘤的新型C-kit T670i突变体选择性激酶抑制剂(GISTS)
机译:发现2-(4-氯-3-(三氟甲基)苯基)-N-(4 - (((6,7-二甲氧基喹啉-4-基)氧基)苯基)乙酰胺(CHMFL-KIT-64),为口服的新颖 用于胃肠道基质肿瘤的C-kit激酶的广谱突变体的可用强化抑制剂
机译:N-((1-(4-(3-(3-((6,7-二甲氧基喹啉-3-基)氧基)苯基)脲基)-2-(三氟甲基)苯基)哌啶-4-基)甲基的发现丙酰胺(CHMFL-KIT-8140)作为能够抑制cKIT激酶T670I“ Gatekeeper”突变体的II型强抑制剂
机译:发现一种用于胃肠道间质瘤(GIST)的高选择性KIT激酶原代V559D突变抑制剂
机译:发现有效的选择性干细胞因子受体/血小板衍生的生长因子受体α(C-KIT / PDGFR)双抑制剂,用于治疗伊马替尼抗性胃肠肿瘤肿瘤(GISTS)