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机译:(r)-6-新戊基-2-(吡啶-2-基甲氧基)-6,7-二氢嘧啶[2,1-c] [1,4]恶化-4(9h)-one(PF- 06462894),缺乏缺乏的代谢性谷氨酸受体5,在大鼠和非人的灵长类动物中分析阴性变形调节剂
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Pharmacokinet Dynam &
Metab Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Res Unit Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Drug Safety Res &
Dev Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Pharmacokinet Dynam &
Metab Groton CT 06340 USA;
Pfizer Inc Biolmaging Ctr Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Pharmaceut Sci Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Drug Safety Res &
Dev Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Pharmaceut Sci Groton CT 06340 USA;
Pfizer Inc Biostat Early Clin Dev Groton CT 06340 USA;
Pfizer Inc Drug Safety Res &
Dev Groton CT 06340 USA;
Pfizer Inc Pharmacokinet Dynam &
Metab Groton CT 06340 USA;
Pfizer Inc Pharmacokinet Dynam &
Metab Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Biolmaging Ctr Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Res Unit Cambridge MA 02139 USA;
Pfizer Inc Pharmacokinet Dynam &
Metab Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Drug Safety Res &
Dev Groton CT 06340 USA;
Pfizer Inc Biolmaging Ctr Groton CT 06340 USA;
Pfizer Inc Neurosci &
Pain Res Unit Cambridge MA 02139 USA;
Pfizer Inc Neurosci &
Pain Med Chem Cambridge MA 02139 USA;
Pfizer Inc Pharmacokinet Dynam &
Metab Cambridge MA 02139 USA;
机译:(r)-6-新戊基-2-(吡啶-2-基甲氧基)-6,7-二氢嘧啶[2,1-c] [1,4]恶化-4(9h)-one(PF- 06462894),缺乏缺乏的代谢性谷氨酸受体5,在大鼠和非人的灵长类动物中分析阴性变形调节剂
机译:代谢型谷氨酸受体2沉默变构调节剂化学转化为双重代谢型谷氨酸受体2/3负/正变构调节剂
机译:1?甲基?3-(4?甲基吡啶?3?基)?6?(吡啶?2?基甲氧基)?1H?吡唑并-[3,4?b]吡嗪(PF470)的发现和临床前表征,选择性和有效的代谢型谷氨酸受体5(mGluR5)负变构调节剂
机译:发现和表征人类alpha4beta2神经元烟碱受体的选择性负变构调节剂。
机译:发现代谢型谷氨酸受体亚型5的6-(嘧啶-5-基甲基)喹啉-8-羧酰胺负变构调节剂
机译:4-氧代1-芳基-1,4-二氢喹啉-3-甲酰胺的设计为代谢谷氨酸受体亚型的选择性阴性变构调节剂2