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机译:新型N-芳基烟酰胺衍生物:服用3,6-二氮杂双环[3.1.1]庚烷作为神经元乙酰胆碱受体的配体
Univ Sassari Dipartimento Chim &
Farm Via F Muroni 23-A I-07100 Sassari Italy;
CNR Inst Neurosci Via Vanvitelli 32 I-20129 Milan Italy;
Univ Sassari Dipartimento Chim &
Farm Via F Muroni 23-A I-07100 Sassari Italy;
Univ Sassari Dipartimento Chim &
Farm Via F Muroni 23-A I-07100 Sassari Italy;
IRCCS Neuromed Via Atinese 18 I-86077 Pozzilli IS Italy;
Sapienza Univ Roma Dipartimento Fisiol &
Farmacol V Erspamer Ple Aldo Moro 5 I-00185 Rome Italy;
IRCCS Neuromed Via Atinese 18 I-86077 Pozzilli IS Italy;
Univ Innsbruck Ctr Mol Biosci CMBI Inst Pharm Pharmacognosy Innrain 80-82 A-6020 Innsbruck;
Univ Milan Dept Med Biotechnol &
Translat Med Milan Italy;
Univ Milan Dept Med Biotechnol &
Translat Med Milan Italy;
Paracelsus Med Univ Salzburg Dept Pharmaceut Chem Salzburg Austria;
Univ Sassari Dipartimento Chim &
Farm Via F Muroni 23-A I-07100 Sassari Italy;
Univ Sassari Dipartimento Chim &
Farm Via F Muroni 23-A I-07100 Sassari Italy;
Univ Sassari Dipartimento Chim &
Farm Via F Muroni 23-A I-07100 Sassari Italy;
3; 6-diazabicyclo3.1.1heptanes; Synthesis; nAChRs; Partial agonists; alpha(4)beta(2) selectivity; Tobacco addiction; Molecular docking;
机译:新型N-芳基烟酰胺衍生物:服用3,6-二氮杂双环[3.1.1]庚烷作为神经元乙酰胆碱受体的配体
机译:具有有效和选择性亲和力的新型3,6-二氮杂双环[3.1.1]庚烷衍生物的设计对α(4)beta(2)神经元烟碱乙酰胆碱受体
机译:鉴定和3,6-二氮杂双环[3.1.1]庚烷-3-羧酰胺作为α4bet2和α6/ alpha3beta2beta3烟碱乙酰胆碱受体(nAChRs)的新型配体
机译:麻醉剂通过神经元烟碱乙酰胆碱受体调节谷氨酸和GABA的释放
机译:脂质双层分子模型嵌入野生型和突变的人M(1)毒蕈碱型乙酰胆碱受体与乙酰胆碱配体。
机译:37-二氮杂双环3.3.1壬烷骨架用于亚型选择性烟碱乙酰胆碱受体配体。第2部分。具有不同间隔基序的羧酰胺衍生物
机译:新型N-芳基烟酰胺衍生物:服用3,6-二氮杂双环3.1.1庚烷作为神经元乙酰胆碱受体的配体