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首页> 外文期刊>Synthetic Communications: An International Journal for Rapid Communication of Synthetic Organic Chemistry >N-Aryl Modification in ?3-Lactam: Design and Synthesis of Novel Monocyclic ?3-Lactam Derivatives as Inhibitor for Bacterial Propagation

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N-Aryl Modification in ?3-Lactam: Design and Synthesis of Novel Monocyclic ?3-Lactam Derivatives as Inhibitor for Bacterial Propagation

机译：α3-内酰胺中的N-芳基修饰：新型单环β3-内酰胺衍生物作为细菌繁殖抑制剂的设计与合成

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《Synthetic Communications: An International Journal for Rapid Communication of Synthetic Organic Chemistry》 |2012年第20期|3031-3041|共11页
作者
Prasanta Patra; Sugata Bhattacharya;
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1. N-aryl modification in-lactam: Design and synthesis of novel monocyclic-lactam derivatives as inhibitor for bacterial propagation [J] . Patra P., Kar G.K., Sarkar A., Synthetic Communications . 2012,第19a21期

机译：N-芳基修饰内酰胺：设计和合成新型单环内酰胺衍生物作为细菌繁殖的抑制剂
2. Design, synthesis and biological evaluation of novel hybrids of N-aryl pyrrothine-base alpha-pyrone as bacterial RNA polymerase inhibitors [J] . Tan Xiangduan, Huang Mohan, Nian Siyun, Bioorganic and Medicinal Chemistry Letters . 2020,第11期

机译：基于芳基丙氨酸碱基α-吡喃酮作为细菌RNA聚合酶抑制剂的设计，合成和生物学评价
3. Discovery of novel bacterial FabH inhibitors (Pyrazol-Benzimidazole amide derivatives): Design, synthesis, bioassay, molecular docking and crystal structure determination [J] . Wang Yan-Ting, Shi Tian-Qi, Fu Jie, European Journal of Medicinal Chemistry: Chimie Therapeutique . 2019,第期

机译：新型细菌FabH抑制剂的发现（吡唑 - 苯并咪唑酰胺衍生物）：设计，合成，生物测定，分子对接和晶体结构测定
4. Quantitative structure-activity relationship (QSAR) modelling of N-aryl derivatives as cholinesterase inhibitors [C] . Ridzuan Mohd Syafiq Mohammad, Jaafar Mohd Zuli, Zain Mazatulikhma Mat 2012 IEEE Symposium on Humanities, Science and Engineering Research . 2012

机译：N-芳基衍生物作为胆碱酯酶抑制剂的定量构效关系（QSAR）模型
5. Part One. Synthesis of optically active tryptophan derivatives with potential activity as indoleamine 2,3-dioxygenase inhibitors: An approach via asymmetric catalytic hydrogenation. Part Two. Design, synthesis and pharmacology of selective ligands for alpha1-containing GABA(A)/benzodiazepine receptor subtypes: SAR studies of beta-carbolines at positions -3 and -6 and their corresponding bivalent ligands. Part Three. First enantiospecific total synthesis of the important biogenetic intermediates, (+)-polyneuridine and (+)-polyneuridine aldehyde, as well as 16-epi-vellosimine and macusine A. [D] . Yin, Wenyuan. 2007

机译：第一部分。具有吲哚胺2,3-二加氧酶抑制剂潜在活性的旋光色氨酸衍生物的合成：一种通过不对称催化氢化的方法。第二部分。含α1的GABA（A）/苯并二氮杂receptor受体亚型的选择性配体的设计，合成和药理作用：位于-3和-6位的β-咔啉及其相应的二价配体的SAR研究。第三部分。重要生物遗传中间体，（+）-聚神经氨酸和（+）-聚神经氨酸醛，以及16-表-维西辛和Macusine A的首次对映体全合成。
6. Design and characterization of N2-arylaminopurines which selectively inhibit replicative DNA synthesis and replication-specific DNA polymerases: guanine derivatives active on mammalian DNA polymerase alpha and bacterial DNA polymerase III. [O] . G E Wright, E F Baril, V M Brown, 1982

机译：N2-芳基氨基嘌呤的设计和表征其选择性抑制复制性DNA合成和复制特异性DNA聚合酶：对哺乳动物DNA聚合酶α和细菌DNA聚合酶III具有活性的鸟嘌呤衍生物。
7. The Rational Design, Synthesis, and Antimicrobial Properties of Thiophene Derivatives That Inhibit Bacterial Histidine Kinases [O] . Boibessot, Thibaut, zschiedrich, Christopher, Lebeau, Alexandre, 2016

机译：抑制细菌组氨酸激酶的噻吩衍生物的合理设计，合成和抗菌性能

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