首页> 外国专利> Acyl Coenzyme A: novel N-aryl and N-heteroaryl urea derivatives as inhibitors of cholesterol acyltransferases (ACAT) (NEW N-ARYL AND N-HETEROARYLUREA DERIVATIVES AS INHIBITORS OF ACYL COYLENE A: CHOLESTEROL ACYL TRANSFERASE (ACAT)

Acyl Coenzyme A: novel N-aryl and N-heteroaryl urea derivatives as inhibitors of cholesterol acyltransferases (ACAT) (NEW N-ARYL AND N-HETEROARYLUREA DERIVATIVES AS INHIBITORS OF ACYL COYLENE A: CHOLESTEROL ACYL TRANSFERASE (ACAT)

机译:酰基辅酶A:新型N-芳基和N-杂芳基脲衍生物作为胆固醇酰基转移酶(ACAT)的抑制剂(作为抑制剂的新的N-芳基和N-杂芳基脲衍生物A:胆固醇酰基转移酶(ACAT)

摘要

The present invention relates to compounds of the general formula (I): RTI ID = 0.0 pharmaceutically /RTI & ;Wherein Q, R17, R18And ROneAre as defined above. The compound of formula (I) above is an inhibitor of acyl-Coenzyme A: cholesterol acyltransferase (ACAT), which is useful as a hyperlipidemic and atherosclerotic agent.
机译:本发明涉及通式(I)的化合物:药学上的;其中Q,R Sup 17,R 18 S和R 一个如上所述。上述式(I)的化合物是酰基辅酶A:胆固醇酰基转移酶(ACAT)的抑制剂,其可用作高脂血症和动脉粥样硬化剂。

著录项

  • 公开/公告号KR950701621A

    专利类型

  • 公开/公告日1995-04-28

    原文格式PDF

  • 申请/专利权人 알렌 제이. 스피겔;

    申请/专利号KR19940704262

  • 发明设计人 어니스트 에스. 하마나카;

    申请日1994-11-26

  • 分类号C07D213/75;A61K31/44;

  • 国家 KR

  • 入库时间 2022-08-22 04:10:43

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